SCHEMBL8560113

SCHEMBL8560113

COc1cc(C(=O)N2c3ccccc3CNc3ccccc32)ccc1NC(=O)c1ccccc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
AVPR2 P30518 5/20 0.44
AVPR1A P37288 5/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44
TUBA1C Q9BQE3 1/20 0.44
TUBB6 Q9BUF5 1/20 0.44
TUBB2B Q9BVA1 1/20 0.44
TUBB1 Q9H4B7 1/20 0.44
AVPR1B P47901 2/20 0.41
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562079 0.91 AVPR2 (0.47) ALDH1A1AVPR2AVPR1ATUBB4ATUBB
SCHEMBL8563485 0.89 PYGL (0.42) ALDH1A1AVPR2AVPR1ATUBB4ATUBB
SCHEMBL8556903 0.86 AVPR2 (0.53) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8562249 0.85 AVPR2 (0.45) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8557684 0.85 AVPR2 (0.51) ALDH1A1AVPR2AVPR1ATUBB4ATUBB
SCHEMBL8559901 0.83 AVPR2 (0.63) AVPR2AVPR1AOXTR
SCHEMBL8557610 0.81 MAPT (0.52) ALDH1A1AVPR2AVPR1APOLBKMT2A
SCHEMBL8557947 0.79 AVPR2 (0.53) AVPR2AVPR1AHPGDOXTR
SCHEMBL8560580 0.77 AVPR2 (0.56) ALDH1A1AVPR2AVPR1AAVPR1BOXTR
SCHEMBL8563394 0.77 NPC1 (0.50) ALDH1A1AVPR2AVPR1AKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed