SCHEMBL8557684

SCHEMBL8557684

COc1cc(C(=O)N2c3ccccc3CNc3ccccc32)ccc1NC(=O)c1ccc(F)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 11/20 0.51
AVPR1A P37288 10/20 0.51
PYGL P06737 4/20 0.50
HTR1F P30939 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40
TUBA1C Q9BQE3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562079 0.89 AVPR2 (0.47) AVPR2AVPR1AALDH1A1TUBB4ATUBB
SCHEMBL8556903 0.87 AVPR2 (0.53) AVPR2AVPR1APYGLKDM4EKMT2A
SCHEMBL8562249 0.86 AVPR2 (0.45) AVPR2AVPR1APYGLKMT2ATUBB4A
SCHEMBL8560113 0.85 ALDH1A1 (0.51) AVPR2AVPR1AALDH1A1KMT2ATUBB4A
SCHEMBL8563485 0.85 PYGL (0.42) AVPR2AVPR1APYGLKDM4EALDH1A1
SCHEMBL8558202 0.81 HTR1F (0.51) AVPR2AVPR1APYGLHTR1F
SCHEMBL8561421 0.80 AVPR2 (0.56) AVPR2AVPR1APYGLHTR1F
SCHEMBL8563279 0.77 AVPR2 (0.48) AVPR2AVPR1AALDH1A1KMT2A
SCHEMBL8561948 0.77 AVPR2 (0.51) AVPR2AVPR1A
SCHEMBL8557610 0.77 MAPT (0.52) AVPR2AVPR1AKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed