SCHEMBL8563463

SCHEMBL8563463

CCCN1CCN(c2cccc3c2ncc2cccn23)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.46
DRD3 P35462 3/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 2/20 0.45
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
ATM Q13315 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTR1A P08908 1/20 0.44
HTR2C P28335 1/20 0.44
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878093 0.83 OPRM1 (0.40) DRD2DRD3KDM4EALDH1A1GAA
SCHEMBL8563995 0.82 DRD2 (0.54) DRD2DRD3KDM4EHTR1AHTR2C
SCHEMBL8572094 0.82 HTR1A (0.48) KDM4EALDH1A1GAAMEN1NPC1
SCHEMBL8563754 0.82 HTR3E (0.53) DRD2DRD3HTR1AHTR2CHTR6
SCHEMBL8569567 0.82 KDM4E (0.47) DRD2KDM4EALDH1A1GAAMEN1
SCHEMBL8570680 0.81 CCR1 (0.39) DRD2DRD3SIGMAR1OPRM1
SCHEMBL8569974 0.81 ALDH1A1 (0.46) DRD2KDM4EALDH1A1GAAMEN1
SCHEMBL8567794 0.80 ALDH1A1 (0.47) DRD3KDM4EALDH1A1GAAMEN1
SCHEMBL8570061 0.80 HTR1A (0.54) DRD2DRD3KDM4EMAPK1HTR1A
SCHEMBL8565559 0.80 DRD4 (0.45) DRD2DRD3KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed