SCHEMBL8564628

SCHEMBL8564628

Cc1ccn2c1cnc1c(N3CCNCC3)cccc12

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.50
HTR2A P28223 2/20 0.49
HTR2C P28335 1/20 0.49
SLC6A4 P31645 1/20 0.49
HTR6 P50406 3/20 0.46
HTR7 P34969 2/20 0.44
HTR1A P08908 5/20 0.44
DRD2 P14416 1/20 0.44
HTR3A P46098 5/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572082 0.86 HTR3E (0.41) HTR2AHTR2CHTR6HTR1ADRD2
SCHEMBL8562645 0.85 DRD2 (0.49) ADRB1HTR2AHTR2CSLC6A4HTR6
SCHEMBL8566442 0.82 ADRB1 (0.33) ADRB1HTR2AHTR2CSLC6A4HTR6
SCHEMBL8569217 0.80 GRM2 (0.44) HTR2AHTR6CYP2C9
SCHEMBL8569105 0.79 DRD2 (0.52) HTR2CHTR6HTR1ADRD2HTR3A
SCHEMBL8564853 0.77 HTR2A (0.45) HTR2AHTR2CSLC6A4HTR6HTR7
SCHEMBL8567130 0.77 HTR1A (0.52) HTR2CHTR6HTR1ADRD2HTR3A
SCHEMBL2532529 0.74 ADRB1 (0.46) ADRB1HTR2AHTR2CSLC6A4HTR6
SCHEMBL19297164 0.74 HTR2A (0.54) ADRB1HTR2AHTR2CSLC6A4HTR6
SCHEMBL8879183 0.74 KDM4E (0.52) HTR2CHTR6HTR7HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed