SCHEMBL8566442

SCHEMBL8566442

Cc1ccn2c1cnc1c(N3CC=CCC3)cccc12

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.33
HTR3E A5X5Y0 2/20 0.32
HTR3B O95264 2/20 0.32
HTR3A P46098 2/20 0.32
HTR3D Q70Z44 2/20 0.32
HTR3C Q8WXA8 2/20 0.32
LCK P06239 1/20 0.32
ESR1 P03372 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
OPRM1 P35372 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
HTR6 P50406 1/20 0.30
CRHR1 P34998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572082 0.82 HTR3E (0.41) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8564628 0.82 ADRB1 (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8572451 0.81 KDM4E (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8569217 0.76 GRM2 (0.44) HTR2AHTR6
SCHEMBL8569105 0.75 DRD2 (0.52) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8567130 0.72 HTR1A (0.52) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7400770 0.70 LCK (0.36) LCK
SCHEMBL8562733 0.68 DRD2 (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8562645 0.68 DRD2 (0.49) ADRB1HTR3AHTR2AHTR2CSLC6A4
SCHEMBL2048248 0.67 ADRB1 (0.53) ADRB1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed