SCHEMBL8565134

SCHEMBL8565134

Clc1ccc(CN2CCN(c3cccc4c3ncc3cccn34)CC2)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.54
HTR2C P28335 4/20 0.54
HTR3E A5X5Y0 5/20 0.53
HTR3B O95264 5/20 0.53
HTR3A P46098 5/20 0.53
HTR3D Q70Z44 5/20 0.53
HTR3C Q8WXA8 5/20 0.53
KDM4E B2RXH2 3/20 0.50
MAPT P10636 1/20 0.50
SIGMAR1 Q99720 1/20 0.46
DRD4 P21917 2/20 0.43
DRD3 P35462 2/20 0.43
ALDH1A1 P00352 2/20 0.42
PLA2G1B P04054 1/20 0.42
RAB9A P51151 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42
CYP2A13 Q16696 1/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566350 0.88 KDM4E (0.52) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL8879183 0.85 KDM4E (0.52) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL8564672 0.83 HTR1A (0.53) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL8563754 0.82 HTR3E (0.53) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL8565559 0.80 DRD4 (0.45) HTR1AKDM4EMAPTDRD4DRD3
SCHEMBL8570061 0.79 HTR1A (0.54) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL8570680 0.77 CCR1 (0.39) SIGMAR1DRD4DRD3
SCHEMBL8563463 0.76 DRD2 (0.46) HTR1AHTR2CKDM4EMAPTSIGMAR1
SCHEMBL8572094 0.76 HTR1A (0.48) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL27666200 0.76 KDM4E (0.60) HTR1AHTR2CHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed