SCHEMBL8566690

SCHEMBL8566690

CN1CCN(C(=O)C(=O)c2ccccc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.62
CHRM1 P11229 2/20 0.62
MAPT P10636 1/20 0.62
POLB P06746 2/20 0.56
KDM4E B2RXH2 2/20 0.54
KMT2A Q03164 1/20 0.54
GAA P10253 1/20 0.52
GRM5 P41594 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
EPHX2 P34913 1/20 0.50
TSHR P16473 1/20 0.49
CYP2C9 P11712 1/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12018338 0.90 CES2 (0.56) HPGDCHRM1MAPTKMT2AGAA
SCHEMBL13875347 0.89 HPGD (0.51) HPGDCHRM1MAPTPOLBKDM4E
SCHEMBL12489727 0.82 HPGD (0.62) HPGDPOLBKMT2AGAACYP2C9
SCHEMBL19380443 0.82 PHGDH (0.66) HPGDCHRM1MAPTPOLBKDM4E
SCHEMBL12018348 0.82 CES2 (0.47) HPGDCHRM1MAPTPOLBKMT2A
SCHEMBL5564719 0.81 HPGD (0.66) HPGDPOLBKMT2AGAACYP2C9
SCHEMBL4143496 0.81 POLB (0.80) HPGDPOLBKMT2AGRM5L3MBTL1
SCHEMBL8382619 0.81 CYP2C19 (0.51) HPGDCHRM1MAPTKMT2AL3MBTL1
SCHEMBL28919752 0.80 MAPT (0.63) MAPTPOLBKMT2ATSHRCYP2C9
SCHEMBL13875346 0.79 ACHE (0.70) HPGDKMT2AGAAGRM5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017077550-A1 A METAL FREE PROCESS FOR THE PREPARATION OF ALPHA-SUBSTITUTED CARBONYL COMPOUNDS FROM ALKENES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2017-05-11 WO claimed
WO-2017077550-A1 A METAL FREE PROCESS FOR THE PREPARATION OF ALPHA-SUBSTITUTED CARBONYL COMPOUNDS FROM ALKENES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2017-05-11 WO disclosed
EP-0596406-B1 Imidazo (1,2-a) Pyridines as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 1998-12-16 EP disclosed