SCHEMBL8566976

SCHEMBL8566976

CC(C)(C)OC(=O)c1ccoc1C=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.34
MAPT P10636 4/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
HTT P42858 1/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HPGD P15428 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL160053 0.81 ADORA2B (0.36) ATRMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL7228617 0.81 ALDH1A1 (0.43) MAPTSMN1; SMN2RAB9AHSD17B10HPGD
SCHEMBL2872850 0.77 TSHR (0.50) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL27718695 0.75 TDP1 (0.36) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL9179871 0.74 ALDH1A1 (0.53) MAPTSMN1; SMN2NPC1RAB9AHTT
SCHEMBL27739732 0.73 CA12 (0.36) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL29952357 0.73 RAB9A (0.42) ATRMAPTSMN1; SMN2NPC1RAB9A
Ethylene SCHEMBL28215210 0.72 CHRM2 (0.36) SMN1; SMN2NPC1RAB9AHTTKMT2A
SCHEMBL9186294 0.71 PKM (0.42) SMN1; SMN2NPC1RAB9AHTTHSD17B10
SCHEMBL7475016 0.70 HSP90AB1 (0.38) MAPTSMN1; SMN2NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed