SCHEMBL856747

SCHEMBL856747

CC(=O)C1Cc2ccccc2C1=O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.56
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 1/20 0.55
MAPT P10636 1/20 0.55
KMT2A Q03164 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
METAP1 P53582 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
TSHR P16473 1/20 0.43
ALDH1A1 P00352 1/20 0.41
CYP19A1 P11511 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23618912 0.84 ACHE (0.55) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL30702212 0.83 MAPT (0.56) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL3948845 0.83 MAPT (0.56) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL29458360 0.82 ACHE (0.53) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL599710 0.82 ACHE (0.53) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL5311960 0.81 KMT2A (0.55) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL1000380 0.81 ACHE (0.51) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL19836626 0.81 ALDH1A1 (0.54) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL6116289 0.81 METAP1 (0.55) ACHEKDM4EMEN1MAPTKMT2A
SCHEMBL29476747 0.81 ACHE (0.51) ACHEKDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111925330-A Preparation method of altimezole 上海阿达玛斯试剂有限公司 2020-11-13 CN claimed
US-11795132-B2 Application of metal hydride/palladium compound system in preparation of 1,3-dicarbonyl compound in cascade reaction of electron-deficient alkene compound SOOCHOW UNIVERSITY (CN) 2023-10-24 US disclosed
US-11795132-B2 Application of metal hydride/palladium compound system in preparation of 1,3-dicarbonyl compound in cascade reaction of electron-deficient alkene compound SOOCHOW UNIVERSITY (CN) 2023-10-24 US disclosed
CN-112458001-B Bacterial strain capable of degrading polycyclic aromatic hydrocarbon and application thereof 上海交通大学 2022-09-27 CN disclosed
US-11180437-B2 Method for preparing 1,3-dicarbonyl compound based on metal hydride/palladium compound system SOOCHOW UNIVERSITY (CN) 2021-11-23 US disclosed
US-20210206707-A1 APPLICATION OF METAL HYDRIDE/PALLADIUM COMPOUND SYSTEM IN PREPARATION OF 1,3-DICARBONYL COMPOUND IN CASCADE REACTION OF ELECTRON-DEFICIENT ALKENE COMPOUND SOOCHOW UNIVERSITY (CN) 2021-07-08 US disclosed
US-20210206708-A1 METHOD FOR PREPARING 1,3-DICARBONYL COMPOUND BASED ON METAL HYDRIDE/PALLADIUM COMPOUND SYSTEM SOOCHOW UNIVERSITY (CN) 2021-07-08 US disclosed
CN-112225700-A Preparation method of altimezole 湖南新合新生物医药有限公司 2021-01-15 CN disclosed
CN-111925330-A Preparation method of altimezole 上海阿达玛斯试剂有限公司 2020-11-13 CN disclosed
CN-111925330-A Preparation method of altimezole 上海阿达玛斯试剂有限公司 2020-11-13 CN disclosed
EP-1280779-B1 NEW POLYCYCLIC INDANYLIMIDAZOLES WITH ALPHA2 ADRENERGIC ACTIVITY ORION CORP (FI) 2005-08-24 EP disclosed
EP-1280779-A1 NEW POLYCYCLIC INDANYLIMIDAZOLES WITH ALPHA2 ADRENERGIC ACTIVITY ORION CORPORATION (FI) 2003-02-05 EP disclosed
US-6362211-B2 FOR THERAPY OF NEUROLOGICAL, PSYCHIATRIC OR COGNITION DISORDER, DIABETES, LIPOLYTIC DISORDER, ORTHOSTATIC HYPOTENSION, OR SEXUAL DYSFUNCTION ORION CORPORATION (FI) 2002-03-26 US disclosed
US-20020013356-A1 New polycyclic indanylimidazoles with alpha2 adrenergic activity ORION CORPORATION (FI) 2002-01-31 US disclosed
WO-2001085698-A1 NEW POLYCYCLIC INDANYLIMIDAZOLES WITH ALPHA2 ADRENERGIC ACTIVITY ORION CORPORATION (FI) 2001-11-15 WO disclosed
EP-0310745-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ORION-YHTYMÄ OY (FI) 1993-01-27 EP disclosed
EP-0183492-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Farmos-Yhtyma Oy (FI) 1989-11-15 EP disclosed
EP-0310745-A2 Substituted imidazole derivatives and their preparation and use ORION-YHTYMÄ OY (FI) 1989-04-12 EP disclosed
US-4689339-A 4-dihydroinden-2-yl-, 4-tetrahydronaphth-2-yl-, and 4-dihydrobenzofuran-2-ylimidazoles, useful to block α2 -adrenergic receptors FARMOS YHTYMA OY (FI) 1987-08-25 US disclosed
EP-0183492-A1 Substituted imidazole derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1986-06-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210206708-A1 METHOD FOR PREPARING 1,3-DICARBONYL COMPOUND BASED ON METAL HYDRIDE/PALLADIUM COMPOUND SYSTEM ODC1, HVCN1, PDCD1 ACHE 3532/4885KDM4E 1311/4885MEN1 1294/4885
US-11180437-B2 Method for preparing 1,3-dicarbonyl compound based on metal hydride/palladium compound system ODC1, HVCN1, PDCD1 ACHE 3532/4885KDM4E 1311/4885MEN1 1294/4885
US-20210206707-A1 APPLICATION OF METAL HYDRIDE/PALLADIUM COMPOUND SYSTEM IN PREPARATION OF 1,3-DICARBONYL COMPOUND IN CASCADE REACTION OF ELECTRON-DEFICIENT ALKENE COMPOUND H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HVCN1, HRH4 ACHE 3399/4885KDM4E 924/4885MEN1 1285/4885
US-20020013356-A1 New polycyclic indanylimidazoles with alpha2 adrenergic activity ADRB2, ADRB1, ADRA1A ACHE 1542/4885KDM4E 4112/4885MEN1 968/4885
US-11795132-B2 Application of metal hydride/palladium compound system in preparation of 1,3-dicarbonyl compound in cascade reaction of electron-deficient alkene compound H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HVCN1, HRH4 ACHE 3399/4885KDM4E 924/4885MEN1 1285/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.