SCHEMBL8567545

SCHEMBL8567545

COc1ccc(C(OC(C)=O)c2cc(Cl)ccc2NC(=O)C(C)(C)C)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.42
TSHR P16473 4/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 6/20 0.42
KMT2A Q03164 6/20 0.42
NPSR1 Q6W5P4 1/20 0.42
LPAR1 Q92633 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566120 0.93 MAPT (0.42) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL8564171 0.89 HSD17B1 (0.46) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL8564973 0.83 LPAR1 (0.43) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL8559172 0.82 ALDH1A1 (0.45) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL14254903 0.74 TSHR (0.68) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL6993599 0.73 KMT2A (0.55) MAPTTSHRALDH1A1KDM4EMEN1
SCHEMBL8979498 0.73 MAPT (0.47) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL8979503 0.73 ALDH1A1 (0.51) MAPTTSHRALDH1A1KDM4EGAA
SCHEMBL4118333 0.73 LPAR1 (0.53) MAPTTSHRALDH1A1KDM4EHPGD
SCHEMBL8560752 0.72 LPAR1 (0.47) ALDH1A1KDM4EGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770438-A CHEMICAL INTERMEDIATES FOR ANTICHOLESTEROL COMPOUNDS, CYCLIZATION TO FORM BENZOXAZEPINE OR BENZOTHIAZEPINE COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed