SCHEMBL8567563

SCHEMBL8567563

O=C1CCN(c2ccc3c(c2)OCCO3)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.45
DRD3 P35462 4/20 0.45
DRD4 P21917 3/20 0.45
CMA1 P23946 1/20 0.44
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CYP11B2 P19099 1/20 0.43
KMT2A Q03164 2/20 0.42
GRK2 P25098 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
PKM P14618 1/20 0.41
PKLR P30613 1/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956979 0.90 DRD2 (0.50) DRD2DRD3DRD4CMA1HTR1A
SCHEMBL1360709 0.80 CMA1 (0.59) CMA1KMT2ANPC1RAB9AALDH1A1
SCHEMBL28686215 0.78 LMNA (0.54) DRD2DRD3DRD4HTR1AADRA2A
SCHEMBL6587606 0.73 ADRB1 (0.59) HTR1AALDH1A1LMNA
SCHEMBL15981860 0.73 DRD2 (0.52) DRD2DRD3DRD4HTR1AADRA2A
SCHEMBL15981859 0.73 DRD2 (0.52) DRD2DRD3DRD4HTR1AADRA2A
SCHEMBL10408416 0.71 ADRB1 (0.51) DRD2DRD4CMA1KMT2ANPC1
SCHEMBL7503757 0.71 TGFBR1 (0.55) DRD2DRD3DRD4HTR1AADRA2A
SCHEMBL9829836 0.71 MAOB (0.36) KMT2AALDH1A1MEN1MAPTKDM4E
SCHEMBL14922286 0.71 SMN1; SMN2 (0.59) DRD2DRD3DRD4HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1223650-A Piperidines and pyrrolidines MERCK PATENT GMBH (DE) 1999-07-21 CN disclosed
EP-0898569-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GmbH (DE) 1999-03-03 EP disclosed
WO-1997040038-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GMBH (DE) 1997-10-30 WO disclosed