SCHEMBL8568607

SCHEMBL8568607

CN(C)C(=O)CC1CCN(C(=O)c2ccc(-c3ccc(C#N)cc3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 1/20 0.49
MKNK1 Q9BUB5 3/20 0.48
MKNK2 Q9HBH9 3/20 0.48
KDM1A O60341 6/20 0.48
SIGMAR1 Q99720 1/20 0.48
EPHX2 P34913 1/20 0.47
ALDH1A1 P00352 1/20 0.47
EGLN1 Q9GZT9 1/20 0.47
CCNK O75909 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
L3MBTL3 Q96JM7 1/20 0.46
GPR119 Q8TDV5 1/20 0.45
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8719948 0.84 KDM1A (0.49) SLC6A7KDM1ASIGMAR1EPHX2ALDH1A1
SCHEMBL8407569 0.84 CCNK (0.51) SLC6A7KDM1ASIGMAR1EPHX2ALDH1A1
SCHEMBL8410754 0.82 ITGB3 (0.54) L3MBTL3
SCHEMBL8430024 0.80 ALDH1A1 (0.56) SLC6A7KDM1ASIGMAR1EPHX2ALDH1A1
SCHEMBL8408016 0.79 SLC6A7 (0.51) SLC6A7MKNK1MKNK2KDM1ASIGMAR1
SCHEMBL16627283 0.77 L3MBTL3 (0.77) SLC6A7MKNK1MKNK2KDM1AEPHX2
SCHEMBL8560134 0.77 KDM1A (0.49) KDM1AEPHX2ALDH1A1EGLN1CCNK
SCHEMBL8244983 0.77 ALDH1A1 (0.56) SLC6A7KDM1ASIGMAR1EPHX2ALDH1A1
SCHEMBL13503971 0.76 GRM5 (0.69) KDM1AEPHX2ALDH1A1L3MBTL3PDK1
SCHEMBL28849726 0.73 EPHX2 (0.51) SLC6A7KDM1ASIGMAR1EPHX2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed