SCHEMBL8569129

SCHEMBL8569129

O=C(c1ccccc1)c1ccccc1NC(=O)C(Cl)(Cl)Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
PDK1 Q15118 1/20 0.52
PDK2 Q15119 1/20 0.52
PDK3 Q15120 1/20 0.52
PDK4 Q16654 1/20 0.52
KMT2A Q03164 3/20 0.51
MAPT P10636 6/20 0.47
HPGD P15428 3/20 0.47
MEN1 O00255 2/20 0.47
HTT P42858 2/20 0.47
MAPK1 P28482 1/20 0.47
AKR1C3 P42330 1/20 0.47
LMNA P02545 1/20 0.47
NPSR1 Q6W5P4 2/20 0.45
PKM P14618 1/20 0.45
TP53 P04637 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
GAA P10253 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083067 0.89 NR4A1 (0.53) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL29118239 0.83 ALDH1A1 (0.58) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL8569299 0.83 MAPT (0.67) ALDH1A1KMT2AMAPTMEN1HTT
SCHEMBL13440495 0.82 TP53 (0.60) ALDH1A1KMT2AMAPTMEN1HTT
SCHEMBL8572049 0.82 KDM4C (0.46) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL6169653 0.81 MEN1 (0.56) ALDH1A1KMT2AHPGDMEN1HTT
SCHEMBL3940689 0.80 ALDH1A1 (0.67) ALDH1A1KMT2AMAPTMEN1AKR1C3
SCHEMBL4678464 0.80 ALDH1A1 (0.67) ALDH1A1KMT2AMAPTMEN1AKR1C3
SCHEMBL3486870 0.80 MAPT (0.49) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL6510419 0.79 PDK1 (0.62) ALDH1A1PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626373-B1 Quinazolinone derivatives SUMITOMO PHARMA (JP) 1998-12-23 EP disclosed
US-5556860-A ANTIISCHEMIC AGENTS, BRAIN DISORDERS AND BLOOD METAL CONCENTRATIONS AND KIDNEY DISEASE SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 1996-09-17 US disclosed
EP-0626373-A1 Quinazolinone derivatives SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1994-11-30 EP disclosed