SCHEMBL8569166

SCHEMBL8569166

COC1=Cc2ccccc2CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.49
KDM1A O60341 1/20 0.42
GPR84 Q9NQS5 1/20 0.39
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
CYP19A1 P11511 1/20 0.39
MAOB P27338 2/20 0.38
NISCH Q9Y2I1 1/20 0.38
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
HRH1 P35367 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30661162 1.00 PTGS2 (0.49) PTGS2KDM1AGPR84CYP11B1CYP11B2
SCHEMBL11025756 0.85 KDM1A (0.46) PTGS2KDM1AGPR84CYP11B1CYP11B2
SCHEMBL8031056 0.81 PTGS2 (0.53) PTGS2GPR84CYP11B1CYP11B2MAOB
SCHEMBL9797964 0.79 CYP11B1 (0.39) PTGS2KDM1AGPR84CYP11B1CYP11B2
SCHEMBL9635350 0.76 KDM1A (0.40) PTGS2KDM1AGPR84CYP11B1CYP11B2
SCHEMBL30661164 0.76 MEN1 (0.39) PTGS2KDM1AGPR84MAOBKDM4E
SCHEMBL9798491 0.76 MEN1 (0.39) PTGS2KDM1AGPR84MAOBKDM4E
SCHEMBL11035078 0.75 CYP11B2 (0.51) PTGS2KDM1ACYP11B1CYP11B2CYP19A1
SCHEMBL8161633 0.75 GPR84 (0.40) PTGS2KDM1AGPR84CYP11B1CYP11B2
SCHEMBL28840682 0.73 ELANE (0.42) PTGS2KDM1AGPR84MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0544488-B1 Substituted phenyl phenol leukotriene antagonists LILLY CO ELI (US) 1998-03-11 EP disclosed
WO-1996036347-A1 USE OF LEUKOTRIENE ANTAGONISTS FOR ALZHEIMER'S DISEASE ELI LILLY AND COMPANY (US) 1996-11-21 WO disclosed
EP-0743064-A1 Leukotriene antagonists for use in the treatment or prevention of alzheimer's disease ELI LILLY AND COMPANY (US) 1996-11-20 EP disclosed
US-5462954-A Antiinflammatory, antiallergens; treating asthma ELI LILLY AND COMPANY (US) 1995-10-31 US disclosed
US-5280034-A Bis-heterocyclic prostaglandin analogs E. R. SQUIBB & SONS, INC. (US) 1994-01-18 US disclosed
EP-0544488-A2 Substituted phenyl phenol leukotriene antagonists ELI LILLY AND COMPANY (US) 1993-06-02 EP disclosed
US-4115216-A QUARTERNARY AMMONIUM COMPOUNDS HOECHST AKTIENGESELLSCHAFT (DE) 1978-09-19 US disclosed