SCHEMBL8583284

SCHEMBL8583284

C=C1SC(=S)N(c2cc(-c3sccc3C)c(O)c(C(C)(C)C)c2)C1=O

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.31
PTGS1 P23219 1/20 0.31
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8582964 0.84 PTGS2 (0.39) PTGS2PTGS1MEN1ALDH1A1GAA
SCHEMBL8579119 0.82 CYP1A2 (0.40) PTGS2PTGS1TDP1MEN1ALDH1A1
SCHEMBL8709022 0.81 FABP4 (0.34) MAPTMAPK1TDP1MEN1ALDH1A1
SCHEMBL8583282 0.77 PTPN1 (0.33) PTGS2
SCHEMBL8583061 0.73 HSPA5 (0.32) PTGS2MEN1ALDH1A1GAAKMT2A
SCHEMBL8911876 0.72 CA2 (0.39) PTGS2PTGS1MAPTTDP1MEN1
SCHEMBL8708475 0.70 PTGS2 (0.40) PTGS2PTGS1MAPTTDP1MEN1
SCHEMBL8496737 0.70 PTGS1 (0.40) PTGS2PTGS1MAPTTDP1MEN1
SCHEMBL9159377 0.68 GABBR2 (0.43) PTGS2PTGS1MAPTMAPK1MEN1
SCHEMBL8306589 0.67 PTGS2 (0.72) PTGS2PTGS1MAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731336-A USING ARYL-SUBSTITUTED RHODAMINES ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed
US-5716975-A NONTOXIC RHODANINE DERIVATIVES; ANTIDIABETIC AGENTS, CATHEPSIN D INHIBITORS, B-AMYLOID PROTEIN REDUCTION ELI LILLY AND COMPANY (US) 1998-02-10 US disclosed