SCHEMBL8587254

SCHEMBL8587254

CCC(C(=O)c1ccc(F)cc1)N1CCCN(c2noc3cc(O)ccc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 10/20 0.45
SLC6A2 P23975 9/20 0.45
DRD2 P14416 4/20 0.45
HTR2A P28223 4/20 0.45
HTR7 P34969 2/20 0.45
KCNH2 Q12809 1/20 0.41
SLC6A4 P31645 7/20 0.40
RAB9A P51151 1/20 0.39
MAPK13 O15264 1/20 0.38
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8588933 0.96 HTR2A (0.47) SLC6A3SLC6A2DRD2HTR2AHTR7
Bromide SCHEMBL8590676 0.95 HTR2A (0.47) SLC6A3SLC6A2DRD2HTR2AHTR7
Hydrochloric Acid SCHEMBL8587433 0.95 HTR2A (0.47) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8590828 0.89 SLC6A3 (0.54) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8589313 0.89 SLC6A2 (0.43) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8589088 0.85 DRD2 (0.45) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8588378 0.84 HTR2A (0.47) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8590493 0.78 SLC6A2 (0.43) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL8590773 0.78 SLC6A2 (0.43) SLC6A3SLC6A2DRD2HTR2AHTR7
SCHEMBL7753903 0.76 ALDH1A1 (0.51) DRD2HTR2AHTR7KCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852022-A Antipsychotic agents, composition and method of use HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1998-12-22 US disclosed
US-5696113-A Antipsychotic agents, compositions and method of use HOECHST MARION ROUSSEL, INC. (US) 1997-12-09 US disclosed