SCHEMBL8588378

SCHEMBL8588378

CC(C(=O)c1ccc(F)cc1)N1CCN(c2noc3cc(O)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.47
DRD2 P14416 5/20 0.47
HTR7 P34969 3/20 0.47
KCNH2 Q12809 1/20 0.43
GRIN2B Q13224 1/20 0.41
CHRNB2 P17787 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
MAPK13 O15264 1/20 0.37
HTR1A P08908 3/20 0.36
HTR1F P30939 1/20 0.36
RAD52 P43351 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8588933 0.87 HTR2A (0.47) HTR2ADRD2HTR7KCNH2SLC6A2
Bromide SCHEMBL8590676 0.86 HTR2A (0.47) HTR2ADRD2HTR7KCNH2SLC6A2
Hydrochloric Acid SCHEMBL8587433 0.86 HTR2A (0.47) HTR2ADRD2HTR7KCNH2SLC6A2
SCHEMBL8590828 0.85 SLC6A3 (0.54) HTR2ADRD2HTR7KCNH2SLC6A2
SCHEMBL8587254 0.84 SLC6A3 (0.45) HTR2ADRD2HTR7KCNH2SLC6A2
SCHEMBL13899001 0.80 KDM4E (0.48) HTR2ADRD2HTR7KCNH2MEN1
SCHEMBL8589313 0.79 SLC6A2 (0.43) HTR2ADRD2HTR7KCNH2SLC6A2
SCHEMBL7753903 0.79 ALDH1A1 (0.51) HTR2ADRD2HTR7KCNH2HTR1A
SCHEMBL7754666 0.78 DRD2 (0.52) HTR2ADRD2HTR7KCNH2HTR1A
SCHEMBL7754509 0.76 DRD2 (0.54) HTR2ADRD2HTR7HTR1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852022-A Antipsychotic agents, composition and method of use HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1998-12-22 US disclosed
US-5696113-A Antipsychotic agents, compositions and method of use HOECHST MARION ROUSSEL, INC. (US) 1997-12-09 US disclosed