SCHEMBL8588933

SCHEMBL8588933

CCC(C(=O)c1ccc(F)cc1)N1CCN(c2noc3cc(O)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.47
DRD2 P14416 6/20 0.47
HTR7 P34969 4/20 0.47
SLC6A2 P23975 3/20 0.43
SLC6A3 Q01959 3/20 0.43
KCNH2 Q12809 2/20 0.43
SLC6A4 P31645 1/20 0.38
RAB9A P51151 1/20 0.37
HTR1A P08908 2/20 0.37
MAPK13 O15264 1/20 0.36
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
LMNA P02545 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8587433 0.99 HTR2A (0.47) HTR2ADRD2HTR7SLC6A2SLC6A3
Bromide SCHEMBL8590676 0.99 HTR2A (0.47) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8587254 0.96 SLC6A3 (0.45) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8590828 0.93 SLC6A3 (0.54) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8589313 0.92 SLC6A2 (0.43) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8589088 0.88 DRD2 (0.45) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8588378 0.87 HTR2A (0.47) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8590773 0.81 SLC6A2 (0.43) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL8590493 0.81 SLC6A2 (0.43) HTR2ADRD2HTR7SLC6A2SLC6A3
SCHEMBL7753903 0.79 ALDH1A1 (0.51) HTR2ADRD2HTR7KCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852022-A Antipsychotic agents, composition and method of use HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1998-12-22 US claimed
US-5852022-A Antipsychotic agents, composition and method of use HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1998-12-22 US disclosed
EP-0833820-A1 BENZISOXAZOLE AND INDAZOLE DERIVATIVES AS ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-04-08 EP disclosed
US-5696113-A Antipsychotic agents, compositions and method of use HOECHST MARION ROUSSEL, INC. (US) 1997-12-09 US disclosed
WO-1996039397-A1 BENZISOXAZOLE AND INDAZOLE DERIVATIVES AS ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-12-12 WO disclosed