SCHEMBL8587396

SCHEMBL8587396

NCC(Cc1cccnc1)NCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 1/20 0.45
VNN1 O95497 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 2/20 0.41
SORT1 Q99523 1/20 0.41
HIF1A Q16665 2/20 0.40
EPAS1 Q99814 2/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GPR132 Q9UNW8 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CHRNA7 P36544 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591111 0.86 GAA (0.47) CYP3A4CYP2C19ALDH1A1NPSR1CYP1A2
SCHEMBL8588407 0.85 LTA4H (0.47) CYP3A4CYP2C19ALDH1A1SMN1; SMN2NPSR1
SCHEMBL8590752 0.83 TSHR (0.45) CYP3A4NAMPTALDH1A1NPSR1CYP1A2
SCHEMBL8588116 0.81 CYP1A2 (0.42) CYP3A4CYP2C19NAMPTALDH1A1CYP1A2
SCHEMBL8590761 0.80 MEN1 (0.50) VNN1CYP3A4NAMPTALDH1A1MAPT
SCHEMBL8589194 0.80 GAA (0.48) CYP3A4CYP2C19NAMPTALDH1A1SMN1; SMN2
SCHEMBL8587389 0.80 ALDH1A1 (0.43) CYP3A4CYP2C19NAMPTALDH1A1MAPT
SCHEMBL8589507 0.78 KIF11 (0.49) ALDH1A1SIGMAR1
SCHEMBL8587466 0.78 KCNH2 (0.56) FFAR2ALDH1A1
SCHEMBL8587669 0.78 CYP2D6 (0.53) CYP3A4NAMPTALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998052890-A1 3-ARYLPROPYLAMINO NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1998-11-26 WO disclosed