SCHEMBL8595488

SCHEMBL8595488

COc1cc2c(cc1Cl)C(C)(C)CC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.50
FTO Q9C0B1 1/20 0.39
AKR1B1 P15121 2/20 0.37
MAPT P10636 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
HSP90AA1 P07900 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
CCR6 P51684 1/20 0.37
CACNA1B Q00975 1/20 0.37
APBA1 Q02410 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL301752 0.86 CA1 (0.44) PGRMAPTALDH1A1CA1CA2
SCHEMBL4233485 0.81 ACHE (0.45) PGRAKR1B1MAPTALDH1A1GAA
SCHEMBL5397188 0.79 PGR (0.43) PGRALDH1A1CA1CA2CA7
SCHEMBL1703338 0.78 RXRA (0.38) PGRFTOMAPTALDH1A1MAPK1
SCHEMBL5400962 0.77 ACHE (0.45) PGRAKR1B1MAPTALDH1A1GAA
SCHEMBL14428501 0.76 TNFSF11 (0.55) PGRMAPTMAPK1CA1CA2
SCHEMBL24524147 0.73 CA1 (0.39) FTOAKR1B1MAPTALDH1A1MAPK1
SCHEMBL6553226 0.73 PDE4B (0.37) PGRMAPTALDH1A1RAB9AGAA
SCHEMBL6554850 0.73 PDE4B (0.37) PGRMAPTALDH1A1RAB9AGAA
SCHEMBL14428500 0.72 PDE4A (0.41) PGRMAPTALDH1A1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed