SCHEMBL8604154

SCHEMBL8604154

CN(C)c1ccc2c(=S)cc[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
AR P10275 2/20 0.39
IP6K1 Q92551 1/20 0.35
ALDH1A1 P00352 8/20 0.34
HSD17B10 Q99714 4/20 0.34
ALOX15 P16050 2/20 0.34
TSHR P16473 1/20 0.34
HPGD P15428 2/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TERT O14746 1/20 0.33
APP P05067 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ELANE P08246 2/20 0.33
GAA P10253 2/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601909 0.83 ALDH1A1 (0.30) ALDH1A1
SCHEMBL8599686 0.81 AR (0.43) KDM4EARALDH1A1HSD17B10ALOX15
SCHEMBL8602948 0.76 RXFP1 (0.52) KDM4EALDH1A1HSD17B10ALOX15HPGD
SCHEMBL8603563 0.75 PARP1 (0.39) KDM4EALDH1A1HSD17B10TSHRCYP3A4
SCHEMBL827584 0.73 AHR (0.50) KDM4EALDH1A1HSD17B10ALOX15TSHR
SCHEMBL31084784 0.73 AHR (0.50) KDM4EALDH1A1HSD17B10ALOX15TSHR
SCHEMBL8604156 0.73 KIF11 (0.47) KDM4EALDH1A1GAAPSMD14
SCHEMBL8084300 0.73 HTR3E (0.45) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL8603706 0.72 TYR (0.53) KDM4EALDH1A1HSD17B10ALOX15HPGD
SCHEMBL22372423 0.72 AR (0.49) KDM4EARIP6K1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773449-A BACTERICIDES FOR HELICOBACTER ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 1998-06-30 US disclosed
EP-0786454-A1 THIOQUINOLONE DERIVATIVE ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1997-07-30 EP disclosed