SCHEMBL8997594

SCHEMBL8997594

C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)Nc1ccccc1Oc1cccc2c1C[C@](NC(=O)OC(C)(C)C)(OC(=O)OCc1ccccc1)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.40
CTSK P43235 3/20 0.37
JAK2 O60674 1/20 0.35
CYP1A2 P05177 5/20 0.35
PSMB5 P28074 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ACHE P22303 1/20 0.34
CYP3A4 P08684 5/20 0.33
CYP2C19 P33261 5/20 0.33
CYP2D6 P10635 4/20 0.33
CYP2C9 P11712 4/20 0.33
ALDH1A1 P00352 3/20 0.33
TSHR P16473 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MME P08473 1/20 0.33
ECE1 P42892 1/20 0.33
LMNA P02545 2/20 0.33
ELANE P08246 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997804 0.93 P2RY1 (0.37) SYKCTSKJAK2CYP1A2CYP3A4
SCHEMBL8997631 0.90 SYK (0.35) SYKCTSKPSMB5CA1CA2
SCHEMBL8997716 0.84 GHSR (0.33) LMNA
SCHEMBL8997612 0.83 SYK (0.41) SYKCTSKCYP1A2PSMB5CA1
SCHEMBL8997810 0.83 P2RY1 (0.39)
SCHEMBL8997648 0.82 SYK (0.38) SYKCA1CA2ACHE
SCHEMBL8997603 0.80 SYK (0.38) SYKCTSKCYP1A2PSMB5CA1
SCHEMBL8575729 0.80 CA1 (0.39) SYKCA1CA2ACHECYP3A4
SCHEMBL8567143 0.80 CA1 (0.39) SYKCA1CA2ACHECYP3A4
SCHEMBL8997699 0.80 CA1 (0.36) SYKCA1CA2ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed