SCHEMBL8997804

SCHEMBL8997804

C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)Nc1cccnc1Oc1cccc2c1C[C@](NC(=O)OC(C)(C)C)(OC(=O)OCc1ccccc1)CC2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 9/20 0.37
SYK P43405 1/20 0.36
JAK2 O60674 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CTSK P43235 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
FNTA P49354 2/20 0.34
FNTB P49356 2/20 0.34
MAPK1 P28482 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC4 P56524 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997594 0.93 SYK (0.40) SYKJAK2CTSKCYP1A2CYP3A4
SCHEMBL8997810 0.91 P2RY1 (0.39) P2RY1KDM4EFNTAFNTBMAPK1
SCHEMBL8997695 0.84 P2RY1 (0.37) P2RY1KDM4EFNTAFNTBMAPK1
SCHEMBL8997628 0.84 CA1 (0.34) P2RY1SYKKDM4ECYP1A2CYP3A4
SCHEMBL8997631 0.83 SYK (0.35) SYKCTSK
SCHEMBL8997778 0.81 MEN1 (0.40) P2RY1SYKKDM4ECYP3A4ALDH1A1
SCHEMBL8997612 0.81 SYK (0.41) SYKCTSKCYP1A2CYP3A4CYP2D6
SCHEMBL8613091 0.79 GHSR (0.40) SYKJAK2CTSKCYP3A4MAPK1
SCHEMBL8997648 0.78 SYK (0.38) SYKHDAC1
SCHEMBL8997603 0.78 SYK (0.38) SYKCTSKCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed