SCHEMBL8615811

SCHEMBL8615811

CCC1(c2c[nH]cn2)Cc2cc(Cl)c([N+](=O)[O-])cc2C1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.38
AKR1B1 P15121 1/20 0.34
ALDH1A1 P00352 3/20 0.33
VCAM1 P19320 5/20 0.32
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8610760 0.86 PGR (0.35) ALDH1A1LMNA
SCHEMBL8613817 0.80 PNMT (0.41) CYP3A4LMNA
SCHEMBL8616157 0.79 ADRA2A (0.36)
SCHEMBL4626063 0.74 ADRA2A (0.40)
SCHEMBL7642900 0.73 ADRA2A (0.40)
Atipamezole SCHEMBL881064 0.71 ADRA2A (0.51) CYP3A4TSHRLMNA
Fipamezole SCHEMBL935549 0.70 ADRA2A (0.57)
SCHEMBL8610304 0.70 ADRA2A (0.40)
Fipamezole SCHEMBL1271449 0.70 ADRA2A (0.57)
Atipamezole SCHEMBL3526769 0.70 ADRA2A (0.50) CYP3A4TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618906-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE JUVANTIA PHARMA LTD OY (FI) 1998-04-22 EP disclosed
US-5498623-A MULTISTAGE REACTION FOR HALOGENATION OF COMPOUNDS, NITRATION, REDUCTION AND CONVERSION TO DIAZONIUM SALT THEN HALOGENATION FOR COGNITIVE DISORDERS ORION-YHTYMA OY (FI) 1996-03-12 US disclosed