Atipamezole

Atipamezole

SCHEMBL881064

CCC1(c2c[nH]cn2)Cc2ccccc2C1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.51
ADRA2B P18089 3/20 0.51
ADRA2C P18825 3/20 0.51
ADRA1B P35368 2/20 0.51
KMT2A Q03164 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
CYP2C19 P33261 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP1A2 P05177 1/20 0.31
PKM P14618 1/20 0.31
NFKB1 P19838 1/20 0.31
THPO P40225 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
LMNA P02545 1/20 0.30
AXL P30530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Atipamezole SCHEMBL3526769 0.98 ADRA2A (0.50) ADRA2AADRA2BADRA2CADRA1BKMT2A
Atipamezole SCHEMBL31147780 0.98 ADRA2A (0.50) ADRA2AADRA2BADRA2CADRA1BKMT2A
SCHEMBL9325632 0.88 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1B
SCHEMBL9325667 0.84 ADRA2A (0.38) ADRA2AADRA2BADRA2CADRA1B
SCHEMBL9325681 0.83 ADRA2A (0.38) ADRA2AADRA2BADRA2CADRA1B
Fipamezole SCHEMBL1271449 0.83 ADRA2A (0.57) ADRA2AADRA2BADRA2CADRA1BAXL
SCHEMBL7642900 0.83 ADRA2A (0.40) ADRA2AADRA2BADRA2CADRA1B
SCHEMBL8610304 0.83 ADRA2A (0.40) ADRA2AADRA2BADRA2CADRA1B
Fipamezole SCHEMBL935549 0.83 ADRA2A (0.57) ADRA2AADRA2BADRA2CADRA1BAXL
Hydrochloric Acid SCHEMBL9325923 0.83 ADRA2A (0.37) ADRA2AADRA2BADRA2CADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 165 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3220942-B1 COMPOSITIONS COMPRISING LOW DOSE DESMOPRESSIN IN COMBINATION WITH AN ALPHA-ADRENERGIC RECEPTOR ANTAGONIST SERENITY PHARMACEUTICALS LLC (US) 2022-04-27 EP claimed
WO-2026042013-A1 MITOCHONDRIAL THERAPY INSTITUTE OF MOLECULAR AND CLINICAL OPHTHALMOLOGY BASEL (IOB) (CH) 2026-02-26 WO disclosed
US-20250381167-A1 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS KIORA PHARMACEUTICALS GMBH (AT) 2025-12-18 US disclosed
EP-4662317-A1 PHARMACEUTICAL COMPOSITION FOR USE IN TREATMENT OF VENOUS THROMBOEMBOLISM Universitetet i Tromsø - Norges Arktiske Universitet (NO) 2025-12-17 EP disclosed
EP-4658639-A1 N,N-DIALKYL-4-(2-ETHYLINDAN-2-YL)-1H-IMIDAZOLE-1-CARBOXAMIDES AND RELATED COMPOUNDS FOR TREATMENT OF NEURODEGENERATIVE DISEASES Univerza V Ljubljani (SI) 2025-12-10 EP disclosed
US-20250354986-A1 AFFINITY ENCODED OSCILLATOR ARRAYS, METHODS, AND RELATED ASPECTS FOR MEASURING MOLECULAR BINDING KINETICS ARIZONA BOARD OF REGENTS ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2025-11-20 US disclosed
US-20250345433-A1 Drug For Treating Disorders Of An Organ Or Tissue Function And Diseases Accompanied By Such Disorders, And The Method For Obtaining It Epshtein, Oleg Iliich (RU) 2025-11-13 US disclosed
US-20250333482-A1 MODULATORS OF MESOTHELIAL ECM MOVEMENT HELMHOLTZ ZENTRUM MUENCHEN DEUTSCHES FORSCHUNGSZENTRUM GESUNDHEIT & UMWELT GMBH (DE) 2025-10-30 US disclosed
US-20250277021-A1 Methods for Preventing and Treating Cardiac Dysfunction and COVID-19 with Activin A Antagonists REGENERON PHARMACEUTICALS, INC. 2025-09-04 US disclosed
US-20250276066-A1 METHODS, COMPOSITIONS AND COMPOUNDS FOR TREATING AGE-RELATED DISEASES AND CONDITIONS GERO PTE LTD (SG) 2025-09-04 US disclosed
EP-0618906-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ANTII SAKARI HAAPALINNA (FI) 1994-10-12 EP disclosed
EP-0589957-A1 USE OF ATIPAMEZOLE FOR THE TREATMENT OF MALE SEXUAL IMPOTENCE. ORION YHTYMAE OY (FI) 1994-04-06 EP disclosed
EP-0372954-B1 Substituted imidazole derivatives and their preparation and use ORION YHTYMAE OY (FI) 1994-03-09 EP disclosed
US-5292887-A Antgonists at postsynoptic adrenoreceptors; hypotensive and antidiabetic agents FARMOS-YHTYMA OY (FI) 1994-03-08 US disclosed
CN-1023219-C Substituted imidazole derivatives and their preparation and use FARMOS OY (FI) 1993-12-22 CN disclosed
WO-1993013074-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Orion-Yhtymä Oy (FI) 1993-07-08 WO disclosed
WO-1992022296-A1 USE OF ATIPAMEZOLE FOR THE TREATMENT OF MALE SEXUAL IMPOTENCE Orion-Yhtymä Oy (FI) 1992-12-23 WO disclosed
WO-1991018886-A1 COMPOUNDS FOR THE TREATMENT OF AGE-RELATED MEMORY IMPAIRMENT AND OTHER COGNITIVE DISORDERS Orion-Yhtymä Oy (FI) 1991-12-12 WO disclosed
CN-1043128-A The imdazole derivatives and the preparation thereof that replace FARMOS OY (FI) 1990-06-20 CN disclosed
EP-0372954-A1 Substituted imidazole derivatives and their preparation and use ORION-YHTYMÀ„ OY (FI) 1990-06-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250276066-A1 METHODS, COMPOSITIONS AND COMPOUNDS FOR TREATING AGE-RELATED DISEASES AND CONDITIONS UPF1, NLN, BRCA1 ADRA2A 3352/4885ADRA2B 3146/4885ADRA2C 3948/4885
US-20250381167-A1 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS DHODH, ALDH1A2, QDPR ADRA2A 1133/4885ADRA2B 856/4885ADRA2C 1204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.