SCHEMBL8615837

SCHEMBL8615837

CN(C)CCN1C(=O)COc2ccc(NC(=O)Nc3ccc(-c4ccncc4)c4ccccc34)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
THRB P10828 1/20 0.39
HTR1D P28221 2/20 0.38
HTR1B P28222 2/20 0.38
HTR1A P08908 1/20 0.38
ROCK2 O75116 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615090 0.76 HTR6 (0.49) HTR1DHTR1BHTR1AMAPTHTR2A
SCHEMBL24170879 0.72 CCR8 (0.47) POLBMAPT
SCHEMBL8615160 0.72 HTR1D (0.64) CYP2D6HTR1DHTR1BROCK2NOS3
SCHEMBL8587765 0.71 HTR1D (0.44) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL8587699 0.71 KDR (0.43) ALDH1A1ROCK2
SCHEMBL8119592 0.70 HTR1A (0.67) HTR1DHTR1BHTR1AMAPTHTR2A
SCHEMBL8588618 0.70 HRH3 (0.41) CYP3A4CYP2D6CYP2C9HTR1DHTR1B
SCHEMBL8657486 0.69 KDM4C (0.38) ALDH1A1HTR1DHTR1BHTR1AROCK2
SCHEMBL8564809 0.69 HTR1D (0.75) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8136744 0.69 HTR1D (0.56) CYP3A4CYP2D6CYP2C9MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998047868-A1 HETEROCYCLE-CONTAINING UREA DERIVATIVES AS 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-10-29 WO disclosed