SCHEMBL8657486

SCHEMBL8657486

CN(C)CCC1CCCc2ccc(NC(=O)Nc3ccc(-c4ccncc4)c4ccccc34)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 6/20 0.38
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
MTNR1A P48039 1/20 0.37
NPC1 O15118 6/20 0.37
RAB9A P51151 5/20 0.37
MCHR1 Q99705 1/20 0.36
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
KDM5B Q9UGL1 3/20 0.34
KDM6B O15054 2/20 0.34
KDM4A O75164 1/20 0.34
KDM4B O94953 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587765 0.72 HTR1D (0.44) HTR1AHTR1DHTR1BNPC1RAB9A
SCHEMBL8587699 0.72 KDR (0.43) MCHR1KMT2AHTR2CHTR2BKDM4E
SCHEMBL8615090 0.72 HTR6 (0.49) HTR1AHTR1DHTR1BNPC1RAB9A
SCHEMBL8588618 0.71 HRH3 (0.41) HTR1DHTR1BMCHR1KMT2AHTR2C
SCHEMBL8130310 0.71 HTR1A (0.44) HTR1AHTR1DHTR1BMEN1KMT2A
SCHEMBL8615837 0.69 POLB (0.39) HTR1AHTR1DHTR1BALDH1A1ROCK2
SCHEMBL6993724 0.68 HTR1D (0.44) HTR1AHTR1DHTR1BNPC1RAB9A
SCHEMBL6999514 0.68 HTR1D (0.59) HTR1AHTR1DHTR1B
SCHEMBL8590672 0.67 KDR (0.45) MCHR1KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL6812318 0.67 MTNR1A (0.67) MTNR1ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998047868-A1 HETEROCYCLE-CONTAINING UREA DERIVATIVES AS 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-10-29 WO disclosed