SCHEMBL8617213

SCHEMBL8617213

CCN1CCN(C2CCC(C(OC)C(=O)O)CC2)C(Nc2ccncc2)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.33
ROCK1 Q13464 4/20 0.33
TRPV6 Q9H1D0 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
CYP3A4 P08684 4/20 0.32
PKN2 Q16513 3/20 0.32
RPS6KA5 O75582 2/20 0.32
LRRK2 Q5S007 2/20 0.32
CYP2D6 P10635 2/20 0.32
TP53 P04637 2/20 0.32
CHUK O15111 1/20 0.32
PRKD3 O94806 1/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
LTK P29376 1/20 0.32
CDK8 P49336 1/20 0.32
PRKX P51817 1/20 0.32
CDK5 Q00535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613339 0.79 KDM4E (0.33) ROCK2ROCK1TRPV6KMT2AMEN1
SCHEMBL8617208 0.74 KDM4E (0.40) ROCK2ROCK1TRPV6KMT2AMEN1
SCHEMBL8617556 0.74 LRRK2 (0.33) LRRK2
SCHEMBL8300408 0.73 KDM4E (0.39) TRPV6KMT2AMEN1CYP2D6CYP1A2
SCHEMBL8612925 0.71 ROCK2 (0.34) ROCK2ROCK1TRPV6KMT2ACYP3A4
SCHEMBL8300207 0.63 CCR2 (0.34) LRRK2
SCHEMBL8616373 0.62 CYP2D6 (0.32) CYP2D6HTTKDM4EALDH1A1
SCHEMBL16785311 0.62
SCHEMBL25872909 0.61 FKBP1A (0.36) MAPTKMT2AMEN1CYP3A4KDM4E
SCHEMBL6026773 0.61 KDM4E (0.56) ROCK2ROCK1MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786371-A INHIBIT AGGREGATION OF BLOOD PLATELETS BOEHRINGER MANNHEIM GMBH (DE) 1998-07-28 US disclosed