SCHEMBL8617546

SCHEMBL8617546

CC(=O)Nc1cccc2c(NC(=N)NC=O)cc(-c3ccccc3C)nc12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PARP14 Q460N5 5/20 0.41
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.38
NUDT1 P36639 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP1A2 P05177 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617040 0.87 KEAP1 (0.41) PARP14HTT
SCHEMBL8616305 0.87 MEN1 (0.36) ALDH1A1SMN1; SMN2HPGDPOLBKDM4E
SCHEMBL8618998 0.87 ABCB1 (0.47) ALDH1A1SMN1; SMN2L3MBTL1HPGDPOLB
SCHEMBL8613400 0.84 GFER (0.41) ALDH1A1SMN1; SMN2HPGDPOLBKDM4E
SCHEMBL8618049 0.84 KDM4E (0.41) ALDH1A1SMN1; SMN2PARP14HPGDPOLB
SCHEMBL8613752 0.82 KMT2A (0.42) ALDH1A1HPGDPOLBKDM4EMAPT
SCHEMBL8613684 0.82 NPC1 (0.42) ALDH1A1SMN1; SMN2HPGDPOLBNUDT1
SCHEMBL8620892 0.82 HTT (0.47) ALDH1A1SMN1; SMN2HPGDPOLBKDM4E
SCHEMBL8615227 0.82 MAPT (0.33) ALDH1A1SMN1; SMN2HPGDPOLBKDM4E
SCHEMBL8617403 0.82 KMT2A (0.41) ALDH1A1L3MBTL1POLBMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed