SCHEMBL8613752

SCHEMBL8613752

CC(=O)Nc1ccc2nc(-c3ccccc3C)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 4/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
PABPC1 P11940 1/20 0.42
RAB9A P51151 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
HTT P42858 1/20 0.40
PDE10A Q9Y233 1/20 0.40
MOK Q9UQ07 4/20 0.39
OPRL1 P41146 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613684 0.92 NPC1 (0.42) KMT2AKDM4EMEN1NPC1MAPT
SCHEMBL8617766 0.88 ABCB1 (0.54) KMT2AKDM4EMEN1NPC1MAPT
SCHEMBL8616047 0.87 ALDH1A1 (0.45) KMT2AKDM4EMAPTRAB9ACA2
SCHEMBL8614948 0.87 HTT (0.39) KMT2AKDM4EMEN1MAPTCA2
SCHEMBL8620892 0.86 HTT (0.47) KMT2AKDM4EMEN1MAPTRAB9A
SCHEMBL8616673 0.84 CA2 (0.50) KMT2AKDM4EMEN1MAPTCA2
SCHEMBL8619083 0.83 CA2 (0.44) KMT2AKDM4EMEN1MAPTRAB9A
SCHEMBL8615234 0.83 HTT (0.38) KMT2AKDM4EMEN1NPC1MAPT
SCHEMBL8618049 0.82 KDM4E (0.41) KMT2AKDM4EMEN1NPC1MAPT
SCHEMBL8617546 0.82 ALDH1A1 (0.41) KMT2AKDM4EMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed