SCHEMBL8617040

SCHEMBL8617040

Cc1ccccc1-c1cc(NC(=N)NC=O)c2cccc(NS(C)(=O)=O)c2n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.41
GLO1 Q04760 3/20 0.40
PLA2G7 Q13093 3/20 0.39
PARP14 Q460N5 2/20 0.36
TP53 P04637 2/20 0.36
NFE2L2 Q16236 1/20 0.36
ALOX15 P16050 1/20 0.36
HTT P42858 1/20 0.36
MMP2 P08253 1/20 0.35
CKS1B P61024 2/20 0.34
SKP2 Q13309 2/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617546 0.87 ALDH1A1 (0.41) PARP14HTT
SCHEMBL8619728 0.87 KEAP1 (0.43) KEAP1GLO1ALOX15HTTMMP2
SCHEMBL8616305 0.86 MEN1 (0.36) PLA2G7TP53ALOX15HTT
SCHEMBL8613761 0.85 TP53 (0.40) KEAP1GLO1PLA2G7TP53NFE2L2
SCHEMBL8613234 0.83 CDK9 (0.38) HTT
SCHEMBL8613400 0.83 GFER (0.41) HTT
SCHEMBL8616047 0.83 ALDH1A1 (0.45) TP53HTT
SCHEMBL8617771 0.83 ALDH1A1 (0.40) TP53HTT
SCHEMBL8613368 0.82 CDK9 (0.38) TP53HTT
SCHEMBL8620892 0.81 HTT (0.47) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed