SCHEMBL8618955

SCHEMBL8618955

N=C(NC=O)Nc1cc(-c2ccccc2)nc2cccc(NS(=O)(=O)C3CCC3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.41
ACP1 P24666 5/20 0.35
ADORA1 P30542 4/20 0.35
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
ADORA3 P0DMS8 2/20 0.34
ADORA2A P29274 2/20 0.34
ABCB1 P08183 1/20 0.34
ABCC1 P33527 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
MEN1 O00255 1/20 0.33
GFER P55789 1/20 0.33
KMT2A Q03164 1/20 0.33
MRGPRX1 Q96LB2 2/20 0.33
CTPS1 P17812 1/20 0.33
GAK O14976 1/20 0.32
STK16 O75716 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
BMP2K Q9NSY1 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617822 0.97 ACLY (0.38) ACLYACP1ADORA1ALOX5APFEN1
SCHEMBL8615331 0.87 ALDH1A1 (0.41) ACP1ABCB1ABCC1ABCG2MEN1
SCHEMBL8614953 0.83 ALDH1A1 (0.42) ACP1ADORA1ADORA3ADORA2AABCB1
SCHEMBL8613211 0.82 ADORA1 (0.38) ACP1ADORA1ADORA3ADORA2AABCB1
SCHEMBL8620212 0.81 SGK1 (0.38) ACLYACP1ADORA1ADORA3ADORA2A
SCHEMBL8615265 0.79 MRGPRX1 (0.37) ACP1ADORA1ABCB1ABCC1ABCG2
SCHEMBL8614064 0.79 ABCB1 (0.50) ACP1ADORA1ADORA3ADORA2AABCB1
SCHEMBL8617724 0.78 ABCG2 (0.41) ACP1ABCB1ABCC1ABCG2MEN1
SCHEMBL8616263 0.77 ABCB1 (0.40) ACP1ADORA1ABCB1ABCC1ABCG2
SCHEMBL8616598 0.77 ABCG2 (0.40) ACP1ABCB1ABCC1ABCG2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed