SCHEMBL8617822

SCHEMBL8617822

N=C(NC=O)Nc1cc(-c2ccccc2)nc2cccc(NS(=O)(=O)C3CCCCC3)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.38
ADORA1 P30542 5/20 0.36
PGAM1 P18669 1/20 0.35
ACP1 P24666 5/20 0.35
ADORA2A P29274 3/20 0.35
ADORA3 P0DMS8 2/20 0.34
PIK3CG P48736 1/20 0.34
DHODH Q02127 1/20 0.33
ABCB1 P08183 1/20 0.33
ABCC1 P33527 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.32
GFER P55789 1/20 0.32
KMT2A Q03164 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
CTPS1 P17812 1/20 0.32
MRGPRX1 Q96LB2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618955 0.97 ACLY (0.41) ACLYADORA1PGAM1ACP1ADORA2A
SCHEMBL8615331 0.86 ALDH1A1 (0.41) ACP1ABCB1ABCC1ABCG2KDM4E
SCHEMBL8614953 0.82 ALDH1A1 (0.42) ADORA1ACP1ADORA2AADORA3ABCB1
SCHEMBL8620212 0.82 SGK1 (0.38) ACLYADORA1ACP1ADORA2AADORA3
SCHEMBL8613211 0.79 ADORA1 (0.38) ADORA1ACP1ADORA2AADORA3DHODH
SCHEMBL8615265 0.79 MRGPRX1 (0.37) ADORA1PGAM1ACP1DHODHABCB1
SCHEMBL8614064 0.78 ABCB1 (0.50) ADORA1ACP1ADORA2AADORA3ABCB1
SCHEMBL8617724 0.77 ABCG2 (0.41) ACP1ABCB1ABCC1ABCG2KDM4E
SCHEMBL8617819 0.77 ACLY (0.42) ACLYDHODHKDM4EMAPTMEN1
SCHEMBL8613362 0.77 ACHE (0.41) ACP1ABCB1ABCC1ABCG2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed