SCHEMBL8630064

SCHEMBL8630064

COC(c1ccccc1F)c1scnc1C

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
P2RX7 Q99572 9/20 0.32
SCN1A P35498 2/20 0.31
SCN5A Q14524 2/20 0.31
SCN8A Q9UQD0 2/20 0.31
SLC6A3 Q01959 1/20 0.31
CTSA P10619 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634186 0.82 MEN1 (0.41) P2RX7MEN1KMT2A
SCHEMBL8629431 0.79 BRD4 (0.39) IDO1TDO2P2RX7
SCHEMBL9025932 0.78 SLC6A3 (0.42) IDO1TDO2SCN1ASCN5ASLC6A3
SCHEMBL28036653 0.72 P2RX7 (0.35) P2RX7SLC6A3CTSA
SCHEMBL8634034 0.72 MEN1 (0.32) P2RX7MEN1KMT2A
SCHEMBL8629520 0.69 ACHE (0.44) IDO1TDO2
SCHEMBL8633317 0.68 ALOX5 (0.31)
SCHEMBL9026067 0.67 SLC6A2 (0.38) IDO1TDO2P2RX7SLC6A3
SCHEMBL28763013 0.66 IDO1 (0.41) IDO1TDO2SLC6A3MEN1KMT2A
SCHEMBL8629570 0.66 GAA (0.44) IDO1TDO2P2RX7SLC6A3CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed