SCHEMBL8630170

SCHEMBL8630170

O=S(=O)(Nc1nn(Cc2ccccc2)c(C(F)(F)F)c1-c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.43
EDNRB P24530 1/20 0.42
EDNRA P25101 1/20 0.42
PTGS2 P35354 1/20 0.41
PPARG P37231 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SERPINE1 P05121 1/20 0.38
CDC25A P30304 1/20 0.38
CDC25B P30305 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KMT2A Q03164 1/20 0.38
LIMK2 P53671 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629982 0.93 EDNRB (0.43) CDC7EDNRBEDNRAPTGS2PTGDR2
SCHEMBL8635531 0.93 PTGS2 (0.50) CDC7EDNRBEDNRAPTGS2PTGDR2
SCHEMBL8629928 0.92 PTGS2 (0.43) CDC7PTGS2PTGDR2SMN1; SMN2KDM4E
SCHEMBL8629382 0.90 ALDH1A1 (0.41) CDC7EDNRBEDNRAPTGS2PTGDR2
SCHEMBL8631438 0.90 CYP1A2 (0.46) PTGS2PPARGPTGDR2SMN1; SMN2KMT2A
SCHEMBL8632875 0.87 SMN1; SMN2 (0.50) EDNRBEDNRAPTGS2PPARGSMN1; SMN2
SCHEMBL8630525 0.86 CCR4 (0.41) CDC7PTGS2PTGDR2SERPINE1SMN1; SMN2
SCHEMBL8632871 0.86 MAPT (0.42) CDC7PTGS2PPARGPTGDR2CDC25A
SCHEMBL8631859 0.85 KDM1A (0.41) CDC7EDNRBEDNRAPTGDR2SMN1; SMN2
SCHEMBL8628839 0.84 EDNRB (0.41) EDNRBEDNRAPTGS2PPARGKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed