SCHEMBL8630595

SCHEMBL8630595

Cc1ncoc1C(O)c1ccc(F)cc1F

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
HDAC6 Q9UBN7 2/20 0.34
F2RL1 P55085 7/20 0.33
BRD4 O60885 3/20 0.33
GAA P10253 1/20 0.32
SOS1 Q07889 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629576 0.82 BRD4 (0.44) CES2CES1HDAC6BRD4
SCHEMBL8636185 0.78 BRD4 (0.43) BRD4CREBBP
SCHEMBL3909922 0.73 CES2 (0.55) CES2CES1
SCHEMBL8634802 0.73 ALDH1A1 (0.38)
SCHEMBL8632301 0.72 GAA (0.44) BRD4GAA
SCHEMBL8632971 0.71 NOTUM (0.38) GAA
SCHEMBL9026125 0.69 BRD4 (0.36) BRD4CREBBP
SCHEMBL8633722 0.68 BRD4 (0.41) BRD4CREBBP
SCHEMBL8634779 0.67 KMT2A (0.38)
SCHEMBL8634032 0.67 IMPDH2 (0.39) BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed