SCHEMBL8633722

SCHEMBL8633722

Cc1ccc(C(O)c2ocnc2C)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.41
MLKL Q8NB16 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
NOTUM Q6P988 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ACHE P22303 1/20 0.32
CREBBP Q92793 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636185 0.86 BRD4 (0.43) BRD4CYP3A4CYP2C19KMT2ANOTUM
SCHEMBL8634032 0.80 IMPDH2 (0.39) BRD4LMNATSHRHSD17B10ACHE
SCHEMBL9026125 0.76 BRD4 (0.36) BRD4KMT2ACREBBP
SCHEMBL9026465 0.75 ALDH1A1 (0.39) BRD4LMNATSHRHSD17B10CREBBP
SCHEMBL8634779 0.74 KMT2A (0.38) CYP2C19KMT2ALMNAHSD17B10ALDH1A1
SCHEMBL8632301 0.72 GAA (0.44) BRD4LMNATSHRHSD17B10ALDH1A1
SCHEMBL96180 0.71 ACHE (0.50) BRD4MLKLCYP3A4CYP2D6CYP2C19
SCHEMBL8629576 0.70 BRD4 (0.44) BRD4CYP3A4NOTUMACHEALDH1A1
SCHEMBL8634802 0.70 ALDH1A1 (0.38) CYP2D6CYP2C19NOTUMLMNATSHR
Hydrochloric Acid SCHEMBL29699724 0.69 ACHE (0.47) BRD4MLKLCYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed