SCHEMBL8630666

SCHEMBL8630666

CCCC(=O)Oc1ccc(N2CCN(c3ccncc3)CC2)cc1CCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
ALOX15 P16050 1/20 0.41
KHK P50053 2/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
CHRM1 P11229 1/20 0.39
F10 P00742 1/20 0.38
AOC3 Q16853 2/20 0.38
ROCK2 O75116 1/20 0.38
CYP17A1 P05093 1/20 0.38
CYP21A2 P08686 1/20 0.38
CYP11B1 P15538 1/20 0.38
HRH3 Q9Y5N1 3/20 0.38
SPHK1 Q9NYA1 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635347 0.86 ITGB3 (0.44) ITGB3ITGA2BALOX15KHKALDH1A1
SCHEMBL8631347 0.81 MAPT (0.47) ITGB3ITGA2BALDH1A1GAA
SCHEMBL8888301 0.81 ITGB3 (0.45) ITGB3ITGA2BF10HRH3HTR1A
SCHEMBL9079517 0.81 HTR1A (0.41) ITGB3ITGA2BF10CYP17A1CYP21A2
SCHEMBL8635350 0.77 HTR1A (0.41) ITGB3ITGA2BKHKALDH1A1GAA
SCHEMBL7327708 0.76 KHK (0.43) ITGB3ITGA2BALOX15KHKALDH1A1
SCHEMBL8635008 0.74 ITGB3 (0.44) ITGB3ITGA2BALDH1A1GAACHRM1
SCHEMBL8631350 0.73 MAPT (0.46) ALDH1A1GAA
Hydrochloric Acid SCHEMBL8837976 0.73 ITGB3 (0.43) ITGB3ITGA2BALDH1A1GAACHRM1
SCHEMBL8605444 0.69 HRH3 (0.56) ITGB3ITGA2BHRH3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed