SCHEMBL8635347

SCHEMBL8635347

CCCC(=O)Oc1ccc(N2CCN(c3ccncc3)CC2)cc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
ALOX15 P16050 1/20 0.42
HTR1A P08908 2/20 0.42
HTR2A P28223 1/20 0.42
KHK P50053 3/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 1/20 0.40
AOC3 Q16853 2/20 0.39
CYP17A1 P05093 2/20 0.39
CYP21A2 P08686 2/20 0.39
CYP11B1 P15538 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ACHE P22303 1/20 0.38
GRIN2B Q13224 1/20 0.38
P2RX7 Q99572 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635350 0.88 HTR1A (0.41) ITGB3ITGA2BHTR1AHTR2AKHK
SCHEMBL8630666 0.86 ITGB3 (0.42) ITGB3ITGA2BALOX15HTR1AHTR2A
SCHEMBL8631347 0.83 MAPT (0.47) ITGB3ITGA2BGAAALDH1A1MAPT
SCHEMBL8889153 0.80 KDM4E (0.47) ITGB3ITGA2BHTR1AHTR2AALDH1A1
SCHEMBL7400703 0.78 KDM4E (0.49) ITGB3ITGA2BALOX15HTR1AHTR2A
SCHEMBL8635008 0.76 ITGB3 (0.44) ITGB3ITGA2BGAAALDH1A1HRH3
SCHEMBL8631350 0.75 MAPT (0.46) GAAALDH1A1MAPT
Hydrochloric Acid SCHEMBL8837976 0.75 ITGB3 (0.43) ITGB3ITGA2BGAAALDH1A1AOC3
SCHEMBL9079517 0.72 HTR1A (0.41) ITGB3ITGA2BHTR1AHTR2ACYP17A1
SCHEMBL9080410 0.71 HRH3 (0.50) HTR1AHTR2AHRH3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed