SCHEMBL8630823

SCHEMBL8630823

COC(=O)c1cc(S(C)(=O)=O)c(N2CCCCC2)cc1C

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
SLC9A1 P19634 2/20 0.47
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.44
CDC25A P30304 1/20 0.40
CDC25B P30305 1/20 0.40
GAA P10253 1/20 0.40
SLC9A3 P48764 1/20 0.40
SLC9A2 Q9UBY0 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705825 0.99 KDM4E (0.48) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL8699987 0.86 SLC6A9 (0.46) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL8700566 0.86 KDM4E (0.55) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL8705791 0.85 KDM4E (0.45) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL8700175 0.85 KDM4E (0.36) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL7158966 0.83 SLC9A1 (0.48) SMN1; SMN2SLC9A1ALDH1A1LMNATSHR
SCHEMBL8635738 0.82 SLC9A1 (0.47) SLC9A1ALDH1A1TSHRSLC9A3SLC9A2
SCHEMBL9259719 0.80 CKS1B (0.41)
SCHEMBL2976531 0.79 PIK3C3 (0.39) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL7764853 0.79 SLC9A1 (0.69) SLC9A1SLC9A3SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753680-A Heterocyclyl-benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-19 US disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed