SCHEMBL8632107

SCHEMBL8632107

Cc1cc(Nc2cccc(C(F)(F)F)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.52
AKR1C2 P52895 2/20 0.52
MPO P05164 4/20 0.48
YAP1 P46937 1/20 0.48
TEAD4 Q15561 1/20 0.48
TEAD2 Q15562 1/20 0.48
RXFP1 Q9HBX9 4/20 0.47
IDH1 O75874 6/20 0.45
RAPGEF4 Q8WZA2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634356 0.87 AKR1C3 (0.49) AKR1C3AKR1C2IDH1
SCHEMBL8632259 0.87 YAP1 (0.49) AKR1C3AKR1C2MPOYAP1TEAD4
SCHEMBL8632908 0.85 PTGS1 (0.43) IDH1RAPGEF4
SCHEMBL7764123 0.84 SLC9A1 (0.54)
SCHEMBL8635252 0.84 AKR1C3 (0.50) AKR1C3AKR1C2IDH1
SCHEMBL8635463 0.83 AKR1C3 (0.45) AKR1C3AKR1C2
SCHEMBL8637536 0.81 AKR1C3 (0.51) AKR1C3AKR1C2IDH1RAPGEF4
SCHEMBL8634318 0.80 PDE4B (0.46)
SCHEMBL8630813 0.80 AKR1C3 (0.50) AKR1C3AKR1C2
SCHEMBL8633408 0.79 ALDH1A1 (0.39) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed