SCHEMBL8633130

SCHEMBL8633130

COc1ccc(OC(=O)CCC2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.52
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
HRH4 Q9H3N8 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP1A2 P05177 2/20 0.47
BDKRB1 P46663 1/20 0.45
CYP2C9 P11712 2/20 0.44
CHRM4 P08173 1/20 0.44
LMNA P02545 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KLK7 P49862 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637465 0.77 CYP2C9 (0.45) F10ALDH1A1HRH3CYP3A4CYP2D6
SCHEMBL8637208 0.77 F10 (0.49) F10HRH3
Hydrochloric Acid SCHEMBL11078727 0.75 TPSAB1 (0.44) F10ALDH1A1SMN1; SMN2KLK7
SCHEMBL7394932 0.75 HRH3 (0.47) F10ALDH1A1GAAHRH3LMNA
SCHEMBL8636538 0.75 F10 (0.44) F10ALDH1A1GAA
SCHEMBL6211789 0.74 POLB (0.61) F10ALDH1A1GAAHRH3CYP3A4
SCHEMBL9409461 0.73 DRD2 (0.48) F10GAALMNA
SCHEMBL4711656 0.72 ITGB3 (0.54)
SCHEMBL7405501 0.72 F10 (0.49) F10ALDH1A1GAAHRH3LMNA
Hydrochloric Acid SCHEMBL9023569 0.72 HTR7 (0.48) ALDH1A1HRH3CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed