SCHEMBL8633408

SCHEMBL8633408

Cc1cc(Nc2ccc(F)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
TBXA2R P21731 2/20 0.39
IDH1 O75874 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
CMA1 P23946 1/20 0.38
PTPN1 P18031 1/20 0.37
MAPK13 O15264 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631102 0.88 AKR1C3 (0.47) ALDH1A1IDH1
SCHEMBL8635463 0.87 AKR1C3 (0.45) ALDH1A1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8634356 0.86 AKR1C3 (0.49) IDH1RAB9A
SCHEMBL8632908 0.86 PTGS1 (0.43) IDH1PTGS1PTGS2CMA1MAPK13
SCHEMBL8634936 0.85 AKR1C3 (0.48) ALDH1A1IDH1SMN1; SMN2
SCHEMBL8635300 0.85 HTT (0.38) ALDH1A1TBXA2RPTGS1PTGS2
SCHEMBL8635344 0.85 KMT2A (0.36) ALDH1A1PTGS1PTGS2
SCHEMBL8636256 0.84 TBXA2R (0.44) ALDH1A1TBXA2R
SCHEMBL27526953 0.84 RAPGEF4 (0.42) ALDH1A1
SCHEMBL7764096 0.82 SLC9A1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed