SCHEMBL8636256

SCHEMBL8636256

Cc1cc(Nc2ccc(C#N)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 8/20 0.44
BRD4 O60885 1/20 0.38
MCL1 Q07820 1/20 0.38
MERTK Q12866 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TNIK Q9UKE5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634318 0.87 PDE4B (0.46) TBXA2RMCL1ALDH1A1
SCHEMBL8635360 0.86 TBXA2R (0.41) TBXA2RMCL1MERTKALDH1A1
SCHEMBL8631102 0.85 AKR1C3 (0.47) ALDH1A1
SCHEMBL8633408 0.84 ALDH1A1 (0.39) TBXA2RALDH1A1
SCHEMBL8635463 0.84 AKR1C3 (0.45) BRD4ALDH1A1
SCHEMBL7761272 0.83 SLC9A1 (0.57)
SCHEMBL27348370 0.83 VNN1 (0.43)
SCHEMBL8634936 0.82 AKR1C3 (0.48) ALDH1A1
SCHEMBL8635344 0.81 KMT2A (0.36) ALDH1A1
SCHEMBL27526953 0.81 RAPGEF4 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed