SCHEMBL8632908

SCHEMBL8632908

Cc1cc(Nc2cccc(F)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
KCNJ6 P48051 1/20 0.41
KCNJ5 P48544 1/20 0.41
KCNJ3 P48549 1/20 0.41
RAPGEF4 Q8WZA2 1/20 0.41
P2RY4 P51582 1/20 0.39
LMNA P02545 1/20 0.39
CNR1 P21554 1/20 0.39
CDC7 O00311 1/20 0.38
DAPK3 O43293 1/20 0.38
PRKD3 O94806 1/20 0.38
PIM1 P11309 1/20 0.38
CDK2 P24941 1/20 0.38
FLT3 P36888 1/20 0.38
CSNK1A1 P48729 1/20 0.38
GSK3B P49841 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
PRKX P51817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635252 0.87 AKR1C3 (0.50) PTGS1PTGS2LMNASMN1; SMN2IDH1
SCHEMBL8633408 0.86 ALDH1A1 (0.39) PTGS1PTGS2SMN1; SMN2CMA1MAPK13
SCHEMBL8635463 0.86 AKR1C3 (0.45) MAPK13MAPK12MAPK11MAPK14MEN1
SCHEMBL8632359 0.86 MEN1 (0.44) PTGS1PTGS2KCNJ6KCNJ5KCNJ3
SCHEMBL8632107 0.85 AKR1C3 (0.52) RAPGEF4IDH1
SCHEMBL8637536 0.84 AKR1C3 (0.51) PTGS1RAPGEF4LMNASMN1; SMN2IDH1
SCHEMBL7766528 0.83 SLC9A1 (0.57)
SCHEMBL8634318 0.83 PDE4B (0.46) PTGS1PTGS2KCNJ6KCNJ5KCNJ3
SCHEMBL8631388 0.81 GAA (0.40) KCNJ6KCNJ5KCNJ3JAK3SMN1; SMN2
SCHEMBL8631102 0.80 AKR1C3 (0.47) KCNJ6KCNJ5KCNJ3LMNAIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed