SCHEMBL8633810

SCHEMBL8633810

Cc1nc(C)c(C(O)c2ccccc2Cl)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGFBP3 P17936 1/20 0.36
ADRB2 P07550 2/20 0.36
ADRB1 P08588 2/20 0.36
AOC3 Q16853 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
CYP2D6 P10635 2/20 0.36
NFKB1 P19838 1/20 0.36
HIF1A Q16665 1/20 0.36
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
GRM4 Q14833 1/20 0.35
BLM P54132 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CASP1 P29466 1/20 0.35
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633796 0.75 ADRB2 (0.36) IGFBP3ADRB2ADRB1AOC3IDO1
SCHEMBL230382 0.71 ADRB2 (0.48) IGFBP3ADRB2ADRB1AOC3IDO1
SCHEMBL29976363 0.71 ADRB2 (0.48) IGFBP3ADRB2ADRB1AOC3IDO1
SCHEMBL22927657 0.66 GAA (0.41) ADRB2ADRB1AOC3CYP2D6NFKB1
SCHEMBL8634802 0.66 ALDH1A1 (0.38) IGFBP3ADRB2ADRB1AOC3CYP2D6
SCHEMBL10860435 0.66 HPGD (0.62) IDO1TDO2CYP2D6HIF1ARAB9A
SCHEMBL12179243 0.66 LMNA (0.31) RAB9ARECQL
SCHEMBL327675 0.65 COMT (0.43) HPGDHSD17B10KMT2A
SCHEMBL15649374 0.65 RORC (0.33)
SCHEMBL11606505 0.64 TSHR (0.50) ADRB2ADRB1AOC3IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1047169-C (1-phenyl-1-heterocyclyl) methanol and (1-phenyl-1-heterocyclyl) methylamine derivatives ASTRA AB (SE) 1999-12-08 CN claimed
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US claimed
CN-1126991-A Novel (1-phenyl-1-heterocyclyl) methanol and (1-phenyl-1-heterocyclyl) methylamine derivatives ASTRA AB (SE) 1996-07-17 CN claimed
CN-1047169-C (1-phenyl-1-heterocyclyl) methanol and (1-phenyl-1-heterocyclyl) methylamine derivatives ASTRA AB (SE) 1999-12-08 CN disclosed
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
CN-1126991-A Novel (1-phenyl-1-heterocyclyl) methanol and (1-phenyl-1-heterocyclyl) methylamine derivatives ASTRA AB (SE) 1996-07-17 CN disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed