SCHEMBL8633796

SCHEMBL8633796

Cc1ncsc1C(O)c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.36
ADRB1 P08588 2/20 0.36
AOC3 Q16853 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
HIF1A Q16665 1/20 0.36
P2RX7 Q99572 4/20 0.35
CYP2C19 P33261 1/20 0.35
BLM P54132 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CASP1 P29466 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
IGFBP3 P17936 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629570 0.84 GAA (0.44) P2RX7SLC6A3IDO1TDO2
SCHEMBL8633346 0.82 LMNA (0.40) P2RX7
SCHEMBL8629431 0.81 BRD4 (0.39) P2RX7IDO1TDO2
SCHEMBL8629520 0.80 ACHE (0.44) IDO1TDO2
SCHEMBL8630486 0.79 KMT2A (0.46) CYP2C19
SCHEMBL8683323 0.77 KDM4E (0.43) CYP2D6P2RX7CYP2C19SLC6A3
SCHEMBL2593085 0.77 SLC6A3 (0.44) SLC6A3IDO1TDO2
SCHEMBL8633810 0.75 IGFBP3 (0.36) ADRB2ADRB1AOC3CYP2D6NFKB1
SCHEMBL8634063 0.74 FFAR2 (0.38) AOC3
SCHEMBL8631273 0.74 BRD4 (0.41) CYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed