SCHEMBL8634665

SCHEMBL8634665

COC1(CC(N)=O)C(CCc2ccccn2)CCc2cc(Cl)ccc2N1C(=O)c1ccc(NC(=O)c2ccccc2Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 4/20 0.41
AVPR1A P37288 4/20 0.41
GRM4 Q14833 3/20 0.38
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
HSD11B1 P28845 3/20 0.36
F11 P03951 1/20 0.35
PPARG P37231 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
NPY2R P49146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634000 0.87 AVPR1A (0.41) AVPR2AVPR1AHSD11B1
SCHEMBL8632078 0.86 AVPR1A (0.42) AVPR2AVPR1AHSD11B1
SCHEMBL8630006 0.86 AVPR2 (0.42) AVPR2AVPR1AHSD11B1KDM4EGAA
SCHEMBL8635113 0.67 CHRM5 (0.42) AVPR2AVPR1AKDM4E
SCHEMBL8627393 0.67 AVPR1A (0.40) AVPR2AVPR1AHSD11B1
SCHEMBL8627408 0.67 AVPR1A (0.40) AVPR2AVPR1AHSD11B1
SCHEMBL8628617 0.67 AVPR1A (0.40) AVPR2AVPR1A
SCHEMBL8714665 0.67 HSD11B1 (0.43) AVPR2AVPR1AGRM4HSD11B1
SCHEMBL8631000 0.66 AVPR1A (0.39) AVPR2AVPR1AHSD11B1
SCHEMBL8628507 0.66 AVPR1A (0.39) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed