SCHEMBL8635462

SCHEMBL8635462

CCc1cc(Nc2cccnc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.41
ALDH1A1 P00352 2/20 0.39
PTGS1 P23219 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
ALPL P05186 2/20 0.38
SGMS2 Q8NHU3 1/20 0.38
NAMPT P43490 2/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635848 0.86 CYP11B2 (0.46) PDE4BALDH1A1ALPLNAMPTNPC1
SCHEMBL8634502 0.86 PTGS1 (0.38) ALDH1A1PTGS1RAB9ASMN1; SMN2
SCHEMBL8635140 0.86 BCAT2 (0.42) ALDH1A1POLB
SCHEMBL7765590 0.84
SCHEMBL8633209 0.82 MEN1 (0.43) PDE4BALDH1A1PTGS1SMN1; SMN2
SCHEMBL8632359 0.81 MEN1 (0.44) PTGS1RAB9ASMN1; SMN2
SCHEMBL8634357 0.80 TYK2 (0.34)
SCHEMBL8633969 0.80 CNR2 (0.43) PTGS1POLB
SCHEMBL8635300 0.79 HTT (0.38) ALDH1A1PTGS1
SCHEMBL8635178 0.79 AKR1C3 (0.48) PDE4BPTGS1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed