SCHEMBL8635722

SCHEMBL8635722

COc1cccc(Cc2nc(Cl)c(Oc3ccccc3)c(OS(=O)(=O)c3ccc(C(C)C)cn3)n2)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHPS P49366 1/20 0.35
EDNRA P25101 7/20 0.34
NPBWR1 P48145 2/20 0.34
EDNRB P24530 6/20 0.34
CYP1A2 P05177 3/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
ADORA1 P30542 1/20 0.33
USP2 O75604 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
DHFR P00374 1/20 0.33
ATM Q13315 1/20 0.33
BRS3 P32247 1/20 0.33
MCHR1 Q99705 1/20 0.33
PGR P06401 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637899 0.93 DHPS (0.43) DHPSEDNRAEDNRB
SCHEMBL8631708 0.88 DHPS (0.42) DHPSEDNRAEDNRBBRS3
SCHEMBL8635760 0.81 DHPS (0.50) DHPSEDNRAEDNRB
SCHEMBL8638012 0.80 DHPS (0.39) DHPSEDNRAEDNRB
SCHEMBL7851037 0.76 DHPS (0.52) DHPSNPBWR1CYP1A2CYP3A4CYP2C19
SCHEMBL8398732 0.68 EDNRA (0.42) DHPSEDNRAEDNRB
SCHEMBL7850977 0.67 DHPS (0.65) DHPSADORA1TSHR
SCHEMBL7842094 0.65 ADORA1 (0.47) CYP1A2CYP3A4CYP2C19ADORA1CYP2C9
SCHEMBL8398581 0.65 NPBWR1 (0.35) DHPSEDNRANPBWR1EDNRBADORA1
SCHEMBL7852059 0.64 EDNRA (0.65) DHPSEDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837708-A CARDIOVASCULAR DISORDERS OF HYPERTENSION, ISCHEMIA, ANGINA PECTORIS AND VASOSPASMS HOFFMANN-LA ROCHE INC. (US) 1998-11-17 US disclosed